RO88220B - Procedeu pentru prepararea unor derivati de cefalosporina - Google Patents

Procedeu pentru prepararea unor derivati de cefalosporina

Info

Publication number
RO88220B
RO88220B RO114217A RO11421784A RO88220B RO 88220 B RO88220 B RO 88220B RO 114217 A RO114217 A RO 114217A RO 11421784 A RO11421784 A RO 11421784A RO 88220 B RO88220 B RO 88220B
Authority
RO
Romania
Prior art keywords
cefalosporine
preparation
certain derivatives
derivatives
certain
Prior art date
Application number
RO114217A
Other languages
English (en)
Romanian (ro)
Other versions
RO88220A (ro
Inventor
Larry Chris Blaszczak
Stjepan Kukolja
Jan Ross Turner
Original Assignee
Eli Lilly And Company
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Eli Lilly And Company filed Critical Eli Lilly And Company
Publication of RO88220A publication Critical patent/RO88220A/ro
Publication of RO88220B publication Critical patent/RO88220B/ro

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D501/00Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/59Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3 with hetero atoms directly attached in position 3
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/52Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
    • C07D333/54Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
    • C07D333/56Radicals substituted by oxygen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/52Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
    • C07D333/54Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
    • C07D333/60Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
RO114217A 1983-04-12 1984-04-10 Procedeu pentru prepararea unor derivati de cefalosporina RO88220B (ro)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/484,129 US4492693A (en) 1983-04-12 1983-04-12 Benzothienylglycyl cephalosporin derivatives

Publications (2)

Publication Number Publication Date
RO88220A RO88220A (ro) 1985-12-30
RO88220B true RO88220B (ro) 1985-12-31

Family

ID=23922870

Family Applications (1)

Application Number Title Priority Date Filing Date
RO114217A RO88220B (ro) 1983-04-12 1984-04-10 Procedeu pentru prepararea unor derivati de cefalosporina

Country Status (23)

Country Link
US (1) US4492693A (en])
EP (1) EP0122154A3 (en])
JP (1) JPS59199692A (en])
KR (1) KR840008654A (en])
AU (1) AU2673684A (en])
CA (1) CA1212938A (en])
CS (1) CS243485B2 (en])
DD (1) DD213927A5 (en])
DK (1) DK187384A (en])
ES (1) ES8600308A1 (en])
FI (1) FI841437A7 (en])
GB (1) GB2137995A (en])
GR (1) GR79908B (en])
GT (1) GT198400056A (en])
IL (1) IL71497A0 (en])
MA (1) MA20093A1 (en])
NO (1) NO841441L (en])
OA (1) OA07701A (en])
PL (1) PL247170A1 (en])
PT (1) PT78403A (en])
RO (1) RO88220B (en])
ZA (1) ZA842694B (en])
ZW (1) ZW4384A1 (en])

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4581352A (en) * 1984-12-03 1986-04-08 Eli Lilly And Company Thienothienylglycyl cephalosporin derivatives
US4692587A (en) * 1986-02-19 1987-09-08 Spirk Jr John W Hand tool and support
EP1451147A4 (en) * 2001-07-24 2007-06-06 Pharmacore Inc AMINO ACID DERIVATIVES
CN103588790A (zh) * 2013-11-29 2014-02-19 中国科学院长春应用化学研究所 7-氨基-3-氯-3-头孢-4-羧酸-对硝基苄基酯的制备方法

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1445685A1 (de) * 1961-09-11 1968-12-05 Lilly Co Eli Antibiotisch wirksame Cephalospransaeurederivate und Verfahren zu ihrer Herstellung
US3560489A (en) * 1966-08-12 1971-02-02 Lilly Co Eli 7-alpha-aminoacyl cephalosporins
US3575969A (en) * 1968-03-04 1971-04-20 Lilly Co Eli Desacetoxycephalosporin antibiotics
US4024133A (en) * 1971-05-14 1977-05-17 Glaxo Laboratories Limited 7β-[2-Etherified oximino-2-(thienyl-,furyl- or pyridylacetamido)]cephalosporins
GB1445979A (en) * 1972-10-25 1976-08-11 Glaxo Lab Ltd Cephalosporin derivatives
GB1399086A (en) * 1971-05-14 1975-06-25 Glaxo Lab Ltd Cephalosporin compounds

Also Published As

Publication number Publication date
EP0122154A2 (en) 1984-10-17
IL71497A0 (en) 1984-07-31
FI841437A0 (fi) 1984-04-11
NO841441L (no) 1984-10-15
CS279584A2 (en) 1985-08-15
CA1212938A (en) 1986-10-21
DK187384A (da) 1984-10-13
PL247170A1 (en) 1985-08-13
FI841437L (fi) 1984-10-13
PT78403A (en) 1984-05-01
DK187384D0 (da) 1984-04-11
MA20093A1 (fr) 1984-12-31
GB8409381D0 (en) 1984-05-23
JPS59199692A (ja) 1984-11-12
KR840008654A (ko) 1984-12-17
US4492693A (en) 1985-01-08
ZA842694B (en) 1985-11-27
ES531531A0 (es) 1985-10-01
ES8600308A1 (es) 1985-10-01
RO88220A (ro) 1985-12-30
GB2137995A (en) 1984-10-17
OA07701A (fr) 1985-08-30
CS243485B2 (en) 1986-06-12
ZW4384A1 (en) 1984-10-03
AU2673684A (en) 1984-10-18
GR79908B (en]) 1984-10-31
GT198400056A (es) 1985-10-03
DD213927A5 (de) 1984-09-26
EP0122154A3 (en) 1985-10-23
FI841437A7 (fi) 1984-10-13

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